Product Overview
CPI-360 | T6810 | TargetMol Chemicals
CAS: 1802175-06-9
Smiles: COc1cc(C)[nH]c(=O)c1CNC(=O)c1c(C)n([C@H](C)C2CCOCC2)c2ccccc12
Formula: C25H31N3O4
Pathway: Apoptosis|||Chromatin/Epigenetic
Target: Apoptosis|||Histone Methyltransferase
Receptor: N/A
Bioactivity: CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
Molecular Weight: 437, 54
