Product Overview
CTOP | TP2052 | TargetMol Chemicals
CAS: 103429-31-8
Smiles:
Formula: C50H67N11O11S2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Potent and selective μ opioid receptor antagonist (Ki values are 0.96 and >10, 000 nM for μ and δ receptors respectively). Causes behavioral effects on central administration in vivo. Also increases K+ currents in rat locus ceruleus neurons in vitro via a μ receptor independent mechanism.
Molecular Weight: 1062, 28
