Product Overview
Etrasimod | TQ0227 | TargetMol Chemicals
CAS: 1206123-37-6
Smiles: OC(=O)C[C@H]1CCc2c1[nH]c1ccc(OCc3ccc(C4CCCC4)c(c3)C(F)(F)F)cc21
Formula: C26H26F3NO3
Pathway: GPCR/G Protein
Target: S1P Receptor|||LPL Receptor
Receptor: N/A
Bioactivity: Etrasimod is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).
Molecular Weight: 457, 493