Product Overview
FLTX1 | T8984 | TargetMol Chemicals
CAS: 1481401-71-1
Smiles: CCC(=C(c1ccccc1)c1ccc(OCCN(C)c2ccc([N+]([O-])=O)c3nonc23)cc1)c1ccccc1
Formula: C31H28N4O4
Pathway: Endocrinology/Hormones
Target: Estrogen Receptor/ERR|||Estrogen/progestogen Receptor
Receptor: N/A
Bioactivity: FLTX1, a fluorescent Tamoxifen derivative that can specifically label intracellular Tamoxifen-binding sites (estrogen receptors) under permeabilized and non-permeabilized conditions. FLTX1 exhibits the potent antiestrogenic properties of Tamoxifen in breast cancer cells. FLTX1 is devoid of the estrogenic agonistic effect on the uterus.
Molecular Weight: 520, 589