Product Overview
MCL0020 | TP1889 | TargetMol Chemicals
CAS: 475498-26-1
Smiles: CC(=O)N[C@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H](Cc1ccc2ccccc2c1)C(N)=O
Formula: C34H39N7O4
Pathway: GPCR/G Protein|||Neuroscience
Target: Melanocortin Receptor
Receptor: N/A
Bioactivity: Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly reverses stress-induced anorexia but has no effect on food intake in free-feeding rats. Exhibits anxiolytic-like activity in vivo.
Molecular Weight: 609, 731