Product Overview
MRTX-1719 | T40254 | TargetMol Chemicals
CAS: 2630904-45-7
Smiles: N#CC1=C(OC2CC2)C=C(Cl)C(F)=C1C3=C(C4=CC5=C(C(NN=C5CN)=O)C=C4)C=NN3C
Formula: C23H18ClFN6O2
Pathway: Chromatin/Epigenetic
Target: Histone Methyltransferase
Receptor: N/A
Bioactivity: MRTX-1719 is a potent first-in-class selective inhibitor of the PRMT5/MTA complex, with an IC 50 of less than 10 nM in PRMT5/MTA MTAP DEL SDMA cells [1] .
Molecular Weight: 464, 88
