Product Overview
(R)-Nepicastat HCl | T6356 | TargetMol Chemicals
CAS: 195881-94-8
Smiles: Cl.NCc1c[nH]c(=S)n1[C@@H]1CCc2c(F)cc(F)cc2C1
Formula: C14H16ClF2N3S
Pathway: Metabolism
Target: Hydroxylase
Receptor: N/A
Bioactivity: (R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
Molecular Weight: 331, 81
