Product Overview
RO 4938581 | T16794 | TargetMol Chemicals
CAS: 883093-10-5
Smiles: FC(F)c1ncn-2c1Cn1ncnc1-c1cc(Br)ccc-21
Formula: C13H8BrF2N5
Pathway: Membrane transporter/Ion channel|||Neuroscience
Target: GABA Receptor
Receptor: N/A
Bioactivity: RO 4938581 is an effective and selective agonist of GABAA α5 inverse (Ki: 4.6 nM for GABAA α5β3γ2a, and shows a lower affinity at α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki, 174, 185, 80 nM, respectively)).
Molecular Weight: 352, 143
