Product Overview
Sparsentan | T5355 | TargetMol Chemicals
CAS: 254740-64-2
Smiles: CCCCC1=NC2(CCCC2)C(=O)N1Cc1ccc(c(COCC)c1)-c1ccccc1S(=O)(=O)Nc1noc(C)c1C
Formula: C32H40N4O5S
Pathway: Endocrinology/Hormones|||GPCR/G Protein
Target: RAAS|||Endothelin Receptor
Receptor: N/A
Bioactivity: Sparsentan is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM, respectively)
Molecular Weight: 592, 76