Product Overview
TIK-301 | T17095 | TargetMol Chemicals
CAS: 118702-11-7
Smiles: COc1cc2c(c[nH]c2cc1Cl)[C@@H](C)CNC(C)=O
Formula: C14H17ClN2O2
Pathway: GPCR/G Protein|||Neuroscience
Target: 5-HT Receptor
Receptor: N/A
Bioactivity: TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM, respectively). TIK-301 is also a 5-HT2B/5-HT2C receptor antagonist with antidepressant action. TIK-301 has the potential for sleep disorders and other circadian rhythm disorders treatment.
Molecular Weight: 280, 75
