Product Overview
TRV-120027 acetate (1234510-46-3 free base) | TP2158L1 | TargetMol Chemicals
CAS: TP2158L1
Smiles: CC(O)=O.C[C@H](C(O)=O)NC([C@H]1N(C([C@H](CC2=CNC=N2)NC([C@H]([C@@H](C)CC)NC([C@H](CC3=CC=C(O)C=C3)NC([C@H](C(C)C)NC([C@H](CCCNC(N)=N)NC(CNC)=O)=O)=O)=O)=O)=O)CCC1)=O
Formula: C45H71N13O12
Pathway: Endocrinology/Hormones
Target: RAAS
Receptor: N/A
Bioactivity: TRV-120027 acetate is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1 receptor) and engages -arrestins while blocking G-protein signaling.
Molecular Weight: 986, 14