Product Overview
VA5 TG2 inhibitor | T29086 | TargetMol Chemicals
CAS: 2088001-24-3
Smiles: O=C(OCC1=CC=CC=C1)N[C@@H](CCCCNC(C=C)=O)C(N2CCN(C(C(C3=O)=CC4=C(O3)C=C(O)C=C4)=O)CC2)=O
Formula: C31H34N4O8
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: VA5 is an transamidase inhibitor by direct binding at the transamidase site. VA5 also inhibits GTP-binding activities. It interaction at the transamidase site locks the protein in the extended/open conformation to disorganize/inactivate the GTP binding/GTPase site.
Molecular Weight: 590, 63
