Product Overview
VPC-13566 | T29111 | TargetMol Chemicals
CAS: 218464-59-6
Smiles: Cc1cccc2c(c[nH]c12)-c1ccc2ccccc2n1
Formula: C18H14N2
Pathway: Endocrinology/Hormones
Target: Androgen Receptor
Receptor: N/A
Bioactivity: VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.
Molecular Weight: 258, 324
