PKCβ inhibitor 1 | T8376

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€452.00 - €1,626.00
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TMC-T8376
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Product Overview

PKCβ inhibitor 1 | T8376 | TargetMol Chemicals

CAS: 257879-35-9

Smiles: O=C1NC(=O)C(=C1Nc1ccccc1)c1cn(CCCn2ccnc2)c2ccccc12

Formula: C24H21N5O2

Pathway: Apoptosis|||Chromatin/Epigenetic|||Cytoskeletal Signaling

Target: Apoptosis|||PKC

Receptor: N/A

Bioactivity: PKCβ inhibitor 1(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2, respectively).

Molecular Weight: 411, 465

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